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Enantioselective catalytic synthesis of α-aryl-α-SCF 3 -β 2,2 -amino acids

Andreas Eitzinger 1 Jean-François Brière 2 Dominique Cahard 2 Mario Waser 1 
1 JKU - Johannes Kepler University Linz [Linz]
2 COBRA - Chimie Organique et Bioorganique : Réactivité et Analyse
Abstract : We herein report a novel entry towards chiral α-SCF3-β2,2-amino acids by carrying out the ammonium salt-catalyzed α-trifluoromethylthiolation of isoxazolidin-5-ones. This approach allowed for high enantioselectivities and high yields and the obtained heterocycles proved to be versatile platforms to access other targets of potential interest.
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Submitted on : Thursday, February 27, 2020 - 3:41:02 PM
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Andreas Eitzinger, Jean-François Brière, Dominique Cahard, Mario Waser. Enantioselective catalytic synthesis of α-aryl-α-SCF 3 -β 2,2 -amino acids. Organic and Biomolecular Chemistry, Royal Society of Chemistry, 2020, 18 (3), pp.405-408. ⟨10.1039/c9ob02666e⟩. ⟨hal-02442629⟩

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