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One-Pot Synthesis of 2,3-Dihydro-pyrrolopyridinones Using in Situ Generated Formimines

Abstract : A novel one-pot methodology is described for the synthesis of functionalized pyrrolopyridinones using in situ generated formimines and an ortho-lithiated pyridinecarboxamide species. Depending on the reaction conditions, this procedure allows versatile access to aminomethylated pyridinecarboxamides, 2,3-dihydro-pyrrolopyridinones, or 1,1-dialkylated 2,3-dihydro-pyrrolopyridinone derivatives.
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https://hal-normandie-univ.archives-ouvertes.fr/hal-02385488
Contributor : Laurent Bischoff <>
Submitted on : Thursday, November 28, 2019 - 6:30:27 PM
Last modification on : Thursday, July 2, 2020 - 3:28:37 AM

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Geoffrey Deguest, Laurent Bischoff. One-Pot Synthesis of 2,3-Dihydro-pyrrolopyridinones Using in Situ Generated Formimines. Organic Letters, American Chemical Society, 2007, 9 (3), pp.545-545. ⟨10.1021/ol063033d⟩. ⟨hal-02385488⟩

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