Oxindole Alkaloids from Neolaugeria Resinosa, Phytochemistry, vol.32, pp.1587-1590, 1993. ,
Isolation of a New Potent Cytotoxic Pigment along with Indigotin from the Pathogenic Basidiomycetous Fungus Schizophyllum commune, Mycopathologia, vol.146, pp.9-12, 1999. ,
Constituents of Trigonostemon chinensis, J. Nat. Prod, vol.73, pp.40-44, 2009. ,
Telescoped Enolate Arylation/HWE Procedure for the Preparation of 3-Alkenyl-Oxindoles: The First Synthesis of Soulieotine, Eur. J. Org. Chem, vol.18, pp.2947-2952, 2009. ,
Total Synthesis of Schizocommunin and Revision of Its Structure, J. Nat. Prod, vol.76, pp.2034-2039, 2013. ,
Oxindole: A chemical prism carrying plethora of therapeutic benefits, Eur. J. Med. Chem, vol.123, pp.858-894, 2016. ,
Identification of a novel 2-oxindole fluorinated derivative as in vivo antitumor agent for prostate cancer acting via AMPK activation ,
Facile synthesis of simple 2-oxindole-based compounds with promising antiproliferative activity, Future Med. Chem, vol.10, pp.269-282, 2018. ,
Spirooxindoles as novel 3D-fragment scaffolds: Synthesis and screening against CYP121 from M. tuberculosis, Bioorg. Med. Chem. Lett, vol.26, pp.3735-3740, 2016. ,
Pyroglutamic sulphonamide as hydrogen-bonding organocatalyst: Enantioselective Diels-Alder cyclization to construct carbazolespirooxindoles, J. Org. Chem, vol.82, pp.6441-6449, 2017. ,
A tunable and enantioselective hetero-Diels-Alder reaction provides access to distinct piperidinoyl spirooxindoles, Angew. Chem. Int. Ed, vol.56, pp.15945-15949, 2017. ,
Push-pull and pull-push effects in isatylidenes, Magn. Reson. Chem, vol.38, pp.172-176, 2000. ,
Palladium-catalyzed asymmetric allylic amination of racemic butadiene monoxide with isatin derivatives, Org. Biomol. Chem, vol.13, pp.5826-5830, 2015. ,
3-Alkenyl-oxindoles: Natural products, pharmaceuticals, and recent synthetic advances in tandem/telescoped approaches, Eur. J. Org. Chem, pp.4527-4547, 2010. ,
Tandem Horner-Wadsworth-Emmons/Heck procedures for the preparation of 3-alkenyl-oxindoles: The synthesis of Semaxanib and GW441756, Tetrahedron, vol.66, pp.6606-6612, 2010. ,
Synthesis of stereodefined 3-alkylideneoxindoles by palladium-catalyzed reactions of 2-(alkynyl)aryl isocyanates with thiols and alcohols, Chem. Lett, vol.38, pp.1174-1175, 2009. ,
Palladium-catalyzed carbonylative annulation reaction of 2-(1-alkynyl)benzenamines: Selective synthesis of 3-(halomethylene)indolin-2-ones, Org. Lett, vol.9, pp.3413-3416, 2007. ,
Oxindole Synthesis by Palladium-catalysed aromatic C-H alkenylation, Chem. Commun, vol.46, pp.2462-2464, 2010. ,
Chemoselective reduction of isatin-derived electron-deficient alkenes using alkylphosphanes as reduction reagents, Eur. J. Org. Chem, vol.14, pp.2668-2672, 2011. ,
Direct regio-, diastereo-, and enantioselective vinylogous Michael Addition of prochiral 3-alkylideneoxindoles to nitroolefins, Adv. Synth. Catal, vol.355, pp.1881-1886, 2013. ,
Room-temperature Palladium-catalyzed intramolecular oxidative aminocarbonylation of vinylic C(sp2)-H Bonds with amines and CO, Eur. J. Org. Chem, vol.3, pp.616-623, 2014. ,
Vinylogous nucleophilic substitution of the hydroxy group in diarylmethanols with 3-propenyl-2-silyloxyindoles: Towards the synthesis of ?-alkylidene-?-diaryl-2-oxindoles, Adv. Synth. Catal, vol.359, pp.1508-1510, 2017. ,
Enantioselective alkylation of 2-oxindoles catalyzed by a bifunctional phase-transfer catalyst: Synthesis of (?)-Debromoflustramine B, Chem. Eur. J, vol.24, pp.4528-4531, 2018. ,
Oxidative conversion of sulfonyl indoles into 3-alkylidene-2-oxindoles under flow chemical conditions, Synthesis, vol.50, pp.371-376, 2018. ,
Synthesis of novel 5-substituted Indirubins as protein kinases inhibitors, Bioorg. Med. Chem, vol.14, pp.6434-6443, 2006. ,
URL : https://hal.archives-ouvertes.fr/hal-00169371
Synthesis of new 4-thiazolidinone-, pyrazoline-, and Isatin-based conjugates with promising antitumor Activity, J. Med. Chem, vol.55, pp.8630-8641, 2012. ,
Synthesis and antiproliferative activity of (Z)-1-Glycosyl-3-(5-oxo-2-thioxoimidazolidin-4-ylidene)indolin-2-ones and (Z)-3-(2-glycosylsulfanyl-4-oxo-4,5-dihydro-thiazol-5-ylidene)indolin-2-Ones, vol.4, pp.10879-10893, 2014. ,
Synthese und reaktionen des 4,5-dichlor-1,2,3-dithiazoliumchlorids, Eur. J. Inorg. Chem, vol.118, pp.1632-1643, 1985. ,
Polysulfur-nitrogen heterocyclic chemistry, J. Heterocycl. Chem, vol.29, pp.639-651, 1992. ,
Comprehensive Heterocyclic Chemistry II I ,
, , vol.6, p.1, 2008.
Synthesis and properties of 1,2,3-dithiazoles, Russ. Chem. Rev, vol.77, pp.521-546, 2008. ,
, -ium chloride, vol.4, pp.3-4, 2009.
The preparation and characterization of 5-substituted-4-chloro-1,2,3-dithiazolium salts and their conversion into 4-substituted-3-chloro-1,2,5-thiadiazoles, Molecules, vol.10, pp.346-359, 2005. ,
5-Dichloro-1,2,3-dithiazolium chloride (Appel salt). Reactions with N-nucleophiles, Tetrahedron, vol.4, pp.10037-10046, 1994. ,
1,2,4-Thiadiazole 4-oxides, Chem. Commun, vol.11, pp.1273-1274, 1996. ,
Reinvestigating the reaction of 1H-pyrazol-5-amines with 4,5-dichloro-1,2,3-dithiazolium chloride: A route to pyrazolo, J. Org. Chem, vol.79, pp.4025-4037, 2014. ,
Antimicrobial and antitumor activity of N-heteroimmine-1,2,3-dithiazoles and their transformation in triazolo-, imidazo-, and pyrazolopirimidines, Bioorg. Med. Chem, vol.10, pp.449-456, 2002. ,
One-Step Conversion of 2-amino-N -arylbenzamidines into 3-aryl-4-imino-3,4-dihydroquinazoline-2-carbonitriles using 4,5-dichloro-1,2,3-dithiazolium chloride, J. Org. Chem, vol.78, pp.9906-9913, 2013. ,
One-Pot Synthesis of 5-phenylimino, 5-thieno or 5-oxo-1,2,3-dithiazoles and evaluation of their antimicrobial and antitumor activity, Bioorg. Med. Chem. Lett, vol.19, pp.136-141, 2009. ,
Synthesis of novel heterocyclic fused pyrimidin-4-one derivatives from imino-1,2,3-dithiazoles, Arkivoc, vol.2017, pp.335-345 ,
New routes to benzothiophenes, isothiazoles and 1,2,3-dithiazoles, J. Chem. Soc. Perkin Trans. 1, vol.22, pp.3345-3349, 1997. ,
Reactions of tetracyanoethylene oxide with 1,2,3-dithiazoles, J. Chem. Soc. Perkin Trans. 1, pp.2505-2509, 1998. ,
Reactions of 1,2,3-dithiazoles with halogenated malononitriles, J. Chem. Soc. Perkin Trans. 1, pp.1236-1241, 2002. ,
The reaction of 4,5-dichloro-1,2,3-dithiazolium chloride with dimethylsulfonium dicyanomethylide: An improved synthesis of (4-chloro-1,2,3-dithiazolylidene)-malononitrile, Tetrahedron, vol.65, pp.6850-6854, 2009. ,
Stereoisomerism in the adducts of Appel salt with activated methylenes, Bull. Soc. Chim. Belg, vol.106, pp.729-730, 1997. ,
New synthesis of isothiazoles from primary enamines, J. Chem. Soc. Perkin Trans. 1, vol.1, pp.77-81, 1998. ,
Synthesis and Reactions of 1,2,3-Dithiazoles. Sulfur Rep, vol.21, pp.147-210, 1998. ,
Novel synthesis and reactions of 5,7-dialkyl-4,6-dioxo-4,5,6,7-tetrahydroisothiazolo[3,4-d]pyrimidine-3-carbonitriles and 6-methyl-4-oxo-4H-1-aza-5-oxa-2-thiaindene-3-carbonitrile, Org. Lett, vol.5, pp.507-510, 2003. ,
Synthesis of new 5-alkylidene-4-chloro-5H-1,2,3-dithiazoles and their stereochemistry, Tetrahedron, vol.55, pp.9651-9667, 1999. ,
The degradation of 4,5-dichloro-1,2,3-dithiazolium chloride in wet solvents, Tetrahedron, vol.65, pp.6859-6862, 2009. ,
New route to 4-alkoxyquinazoline-2-carbonitriles, J. Chem. Soc. Perkin Trans. 1, vol.23, pp.2857-2860, 1996. ,
The Conversion of 2-(4-chloro-5H-1,2,3-dithiazolylideneamino)benzonitriles into 3-aminoindole-2-carbonitriles using triphenylphosphine, Tetrahedron, vol.65, pp.8428-8433, 2009. ,
Synthesis and in vitro antitumour evaluation of benzothiazole-2-carbonitrile derivatives, Eur. J. Med. Chem, vol.34, pp.1053-1060, 1999. ,
Imidazoquinolinethiones from quinolines: A new molecular rearrangement, Chem. Commun, vol.24, pp.2775-2776, 1996. ,
New syntheses of aryl isothiocyanates, J. Chem. Soc. Perkin Trans. 1, vol.5, pp.889-892, 1998. ,
Novel 9-oxo-thiazolo[5,4-f ]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies, Eur. J. Med. Chem, vol.43, pp.1469-1477, 2008. ,
Ring transformation of (4-chloro-5H-1,2,3-dithiazol-5-ylidene)acetonitriles to 3-haloisothiazole-5-carbonitriles, vol.4, pp.7735-7748, 2014. ,
The preparation of dicyano-1,3,4-thiadiazole and tricyanothiazole via 1,2,3-dithiazole chemistry, Tetrahedron, vol.65, pp.9967-9972, 2009. ,
Cyanothioformyl)indoline; a new indoline ring forming reaction, J. Chem. Soc. Perkin Trans. 1, vol.24, pp.4057-4060, 1998. ,
The stereochemistry of 2-oxoindolin-3-ylidene derivatives, J. Heterocycl. Chem, vol.15, pp.633-636, 1978. ,
On the reaction of Isatin with cyanomethylene(triphenyl)-phosphorane. A nucleophilic attack of alkyl phosphites on the carbon-carbon double bond of (E)-oxindolylideneacetonitrile, Tetrahedron, vol.56, pp.1863-1871, 2000. ,
Alkaloids from the root of Isatis Indigotica, J. Nat. Prod, vol.75, pp.1167-1176, 2012. ,
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